Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50036363
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
SmithKline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50026636(17alpha-hydroxy-20alpha-yohimban-16beta-carboxylic...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of rat cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SB46C4PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
SmithKline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of rat cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SB46C4PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
SmithKline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030612((7aR,8S,11aS,12aS)-8-Methyl-5,6,7a,8,11a,12,12a,13...)copy SMILEScopy InChI
Affinity DataKi:  289nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of rat cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SB46C4PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
SmithKline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)copy SMILEScopy InChI
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of rat cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SB46C4PubMed