Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50037727
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50189704(3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobe...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]leuprorelin binding to monkey recombinant LHRH receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ33G8PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50189701(3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobe...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of [125I]leuprorelin binding to monkey recombinant LHRH receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ33G8PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50067485(3-[(Benzyl-methyl-amino)-methyl]-7-(2,6-difluoro-b...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]leuprorelin binding to monkey recombinant LHRH receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ33G8PubMed