Compile Data Set for Download or QSAR
Found 22 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50041652
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)copy SMILEScopy InChI
Affinity DataIC50: 28.2nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412811(CHEMBL458810)copy SMILEScopy InChI
Affinity DataIC50: 32.4nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50084875(8-(2,4-dichlorophenyl)-N-(1,3-dimethoxypropan-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 39.8nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412814(CHEMBL456660)copy SMILEScopy InChI
Affinity DataIC50: 50.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412812(CHEMBL459173)copy SMILEScopy InChI
Affinity DataIC50: 56.2nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412798(EMICERFONT)copy SMILEScopy InChI
Affinity DataIC50: 66.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412809(CHEMBL516170)copy SMILEScopy InChI
Affinity DataIC50: 67.6nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412808(CHEMBL456640)copy SMILEScopy InChI
Affinity DataIC50: 67.6nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412817(CHEMBL464185)copy SMILEScopy InChI
Affinity DataIC50: 89.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412813(CHEMBL513937)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412802(CHEMBL515363)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412799(CHEMBL458599)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412803(CHEMBL456448)copy SMILEScopy InChI
Affinity DataIC50: 145nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412816(CHEMBL464184)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412804(CHEMBL456449)copy SMILEScopy InChI
Affinity DataIC50: 309nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412806(CHEMBL457710)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412815(CHEMBL457742)copy SMILEScopy InChI
Affinity DataIC50: 363nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412810(CHEMBL458626)copy SMILEScopy InChI
Affinity DataIC50: 372nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412800(CHEMBL515532)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412807(CHEMBL457975)copy SMILEScopy InChI
Affinity DataIC50: 1.23E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412801(CHEMBL458600)copy SMILEScopy InChI
Affinity DataIC50: 1.95E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412805(CHEMBL515503)copy SMILEScopy InChI
Affinity DataIC50: 3.24E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C1XPubMed