Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50043664
TargetP2X purinoceptor 7(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50087267((1-(N,O-bis(1,5-isoquinolinesulfonyl)-N-methyl-L-t...)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at recombinant human P2X7 receptor assessed as inhibition of BzATP-mediated Yo-Pro uptake measured for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MQHPubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM85043(CAS_149017-66-3 | CHEMBL69234 | NSC_6093163 | PPAD...)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at recombinant human P2X7 receptor assessed as inhibition of BzATP-mediated Yo-Pro uptake measured for 1 hr by FLIPR assayMore data for this Ligand-Target Pair