Compile Data Set for Download or QSAR
Found 58 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50045314
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056317(CHEMBL3322349)copy SMILEScopy InChI
Affinity DataEC50:  112nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056316(CHEMBL3322348)copy SMILEScopy InChI
Affinity DataEC50:  2.82E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)copy SMILEScopy InChI
Affinity DataEC50:  871nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056319(CHEMBL3322458)copy SMILEScopy InChI
Affinity DataEC50:  1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056320(CHEMBL3322454)copy SMILEScopy InChI
Affinity DataEC50:  1.50E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056321(CHEMBL3322455)copy SMILEScopy InChI
Affinity DataEC50:  4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056322(CHEMBL3322457)copy SMILEScopy InChI
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056323(CHEMBL3322459)copy SMILEScopy InChI
Affinity DataEC50:  9.66E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056324(CHEMBL3322460)copy SMILEScopy InChI
Affinity DataEC50:  8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056325(CHEMBL3322461)copy SMILEScopy InChI
Affinity DataEC50:  8.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056326(CHEMBL3322462)copy SMILEScopy InChI
Affinity DataEC50:  7.60E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056327(CHEMBL3322463)copy SMILEScopy InChI
Affinity DataEC50:  2.43E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056328(CHEMBL3322464)copy SMILEScopy InChI
Affinity DataEC50:  3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056329(CHEMBL3322465)copy SMILEScopy InChI
Affinity DataEC50:  1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056330(CHEMBL3322467)copy SMILEScopy InChI
Affinity DataEC50:  1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056331(CHEMBL3322468)copy SMILEScopy InChI
Affinity DataEC50:  7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056332(CHEMBL3322469)copy SMILEScopy InChI
Affinity DataEC50:  8.85E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)copy SMILEScopy InChI
Affinity DataEC50:  2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056334(CHEMBL3322471)copy SMILEScopy InChI
Affinity DataEC50:  776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056335(CHEMBL3322472)copy SMILEScopy InChI
Affinity DataEC50:  501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056336(CHEMBL3322473)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056337(CHEMBL3322474)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)copy SMILEScopy InChI
Affinity DataEC50:  661nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056339(CHEMBL3322476)copy SMILEScopy InChI
Affinity DataEC50:  123nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056340(CHEMBL3322478)copy SMILEScopy InChI
Affinity DataEC50:  1.62E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056341(CHEMBL3322479)copy SMILEScopy InChI
Affinity DataEC50:  1.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM21279(1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataEC50:  68nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataEC50:  50nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMedDrugBank
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056316(CHEMBL3322348)copy SMILEScopy InChI
Affinity DataEC50:  2.82E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056317(CHEMBL3322349)copy SMILEScopy InChI
Affinity DataEC50:  112nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056318(CHEMBL3322350)copy SMILEScopy InChI
Affinity DataEC50:  3.89E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)copy SMILEScopy InChI
Affinity DataEC50:  871nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056319(CHEMBL3322458)copy SMILEScopy InChI
Affinity DataEC50:  1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056320(CHEMBL3322454)copy SMILEScopy InChI
Affinity DataEC50:  1.51E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056321(CHEMBL3322455)copy SMILEScopy InChI
Affinity DataEC50:  4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056322(CHEMBL3322457)copy SMILEScopy InChI
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056323(CHEMBL3322459)copy SMILEScopy InChI
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056324(CHEMBL3322460)copy SMILEScopy InChI
Affinity DataEC50:  8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056325(CHEMBL3322461)copy SMILEScopy InChI
Affinity DataEC50:  8.51E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056326(CHEMBL3322462)copy SMILEScopy InChI
Affinity DataEC50:  7.59E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056327(CHEMBL3322463)copy SMILEScopy InChI
Affinity DataEC50:  2.40E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056328(CHEMBL3322464)copy SMILEScopy InChI
Affinity DataEC50:  3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056329(CHEMBL3322465)copy SMILEScopy InChI
Affinity DataEC50:  1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056330(CHEMBL3322467)copy SMILEScopy InChI
Affinity DataEC50:  1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056331(CHEMBL3322468)copy SMILEScopy InChI
Affinity DataEC50:  7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056332(CHEMBL3322469)copy SMILEScopy InChI
Affinity DataEC50:  8.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)copy SMILEScopy InChI
Affinity DataEC50:  2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056334(CHEMBL3322471)copy SMILEScopy InChI
Affinity DataEC50:  776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056335(CHEMBL3322472)copy SMILEScopy InChI
Affinity DataEC50:  501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£t W£rzburg

Curated by ChEMBL
LigandPNGBDBM50056336(CHEMBL3322473)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38HVPubMed
Displayed 1 to 50 (of 58 total ) | Next | Last >>
Jump to: