Compile Data Set for Download or QSAR
Found 25 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50046736
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50158983(CHEMBL439883 | E G P P I S I D L S L E L L R K M I...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128760(CHEMBL3628728)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50155967(4-(2-Bromo-4-isopropyl-phenyl)-8-(butyl-ethyl-amin...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128783(CHEMBL3628740)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128764(CHEMBL3628729)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128774(CHEMBL3628730)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128775(CHEMBL3628731)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128786(CHEMBL3628743)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50155974(8-(Butyl-ethyl-amino)-4-(2,4-dichloro-phenyl)-6-me...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128776(CHEMBL3628732)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128777(CHEMBL3628733)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM20973(8-[butyl(ethyl)amino]-4-(4-methoxy-2-methylphenyl)...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128778(CHEMBL3628734)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128780(CHEMBL3628736)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128779(CHEMBL3628735)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128781(CHEMBL3628737)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128782(CHEMBL3628738)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128805(CHEMBL3628744)copy SMILEScopy InChI
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128808(CHEMBL3628854)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128806(CHEMBL3628745)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128785(CHEMBL3628742)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128807(CHEMBL3628746)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128804(CHEMBL3627731)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50128784(CHEMBL3628741)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRF1 receptor expressed in HEK293T cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4MM0PubMed