Compile Data Set for Download or QSAR
Found 21 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50046914
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50412494(CHEMBL452847 | VUF-10497)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50191289(7-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,f]...)copy SMILEScopy InChI
Affinity DataKi:  102nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM26392(2,4-diamino-5,6-disubstituted pyrimidine, 6 | 6-(4...)copy SMILEScopy InChI
Affinity DataKi:  186nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137647(CHEMBL3752085)copy SMILEScopy InChI
Affinity DataKi:  955nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137655(CHEMBL3752270)copy SMILEScopy InChI
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137646(CHEMBL3752195)copy SMILEScopy InChI
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137652(CHEMBL3752225)copy SMILEScopy InChI
Affinity DataKi:  4.27E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137639(CHEMBL3753985)copy SMILEScopy InChI
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137638(CHEMBL3753705)copy SMILEScopy InChI
Affinity DataKi:  7.76E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137651(CHEMBL3753962)copy SMILEScopy InChI
Affinity DataKi:  9.12E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137645(CHEMBL3752383)copy SMILEScopy InChI
Affinity DataKi:  9.77E+3nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137653(CHEMBL3753334)copy SMILEScopy InChI
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137640(CHEMBL3752972)copy SMILEScopy InChI
Affinity DataKi:  1.38E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137650(CHEMBL3752885)copy SMILEScopy InChI
Affinity DataKi:  1.45E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137649(CHEMBL3753621)copy SMILEScopy InChI
Affinity DataKi:  1.51E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137648(CHEMBL3753784)copy SMILEScopy InChI
Affinity DataKi:  1.95E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137654(CHEMBL3754176)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137641(CHEMBL3753967)copy SMILEScopy InChI
Affinity DataKi:  2.63E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137644(CHEMBL3753849)copy SMILEScopy InChI
Affinity DataKi:  3.16E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137642(CHEMBL3752978)copy SMILEScopy InChI
Affinity DataKi:  3.63E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg

Curated by ChEMBL
LigandPNGBDBM50137643(CHEMBL3754008)copy SMILEScopy InChI
Affinity DataKi:  7.24E+4nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03B0KPubMed