Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50047159
TargetB2 bradykinin receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50150940(CHEMBL3774617)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5X8KPubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50146899(4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.410nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5X8KPubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50067281(4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5X8KPubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50146893(4-{(E)-2-[({[2,4-Dichloro-3-(4-ethoxy-2-methyl-qui...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5X8KPubMed