Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50048019
TargetProteasome subunit beta type-8(Mus musculus)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50201035(CHEMBL3907636)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of chymotrypsin like activity of mouse spleen 20S proteasome beta5i subunit using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2417019PubMed
TargetProteasome subunit beta type-8(Mus musculus)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of chymotrypsin like activity of mouse spleen 20S proteasome beta5i subunit using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 15...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Mus musculus)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50201038(CHEMBL3898621)copy SMILEScopy InChI
Affinity DataIC50: 113nMAssay Description:Inhibition of chymotrypsin like activity of mouse spleen 20S proteasome beta5i subunit using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2417019PubMed
TargetProteasome subunit beta type-8(Mus musculus)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50201036(CHEMBL3972546)copy SMILEScopy InChI
Affinity DataIC50: 118nMAssay Description:Inhibition of chymotrypsin like activity of mouse spleen 20S proteasome beta5i subunit using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2417019PubMed
TargetProteasome subunit beta type-8(Mus musculus)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50201037(CHEMBL3978175)copy SMILEScopy InChI
Affinity DataIC50: 483nMAssay Description:Inhibition of chymotrypsin like activity of mouse spleen 20S proteasome beta5i subunit using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2417019PubMed