Found 42 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 7622 TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 1.60nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 2.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 2.40nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 2.60nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 2.90nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 2.90nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
3D Structure (crystal)TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.90nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 3.90nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 4nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 4nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 5.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 5.70nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 6.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 6.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 8.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 8.70nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 9.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 10.4nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 11.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 12.1nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 13.6nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 13.7nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 13.9nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 14.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 15.6nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 15.8nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 15.9nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 35.7nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 39.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 51.8nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 53nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 146nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.
US Patent
Array BioPharma Inc.; Genentech, Inc.
US Patent
Affinity DataIC50: 249nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
