Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 981
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM50023444(CHEMBL3329869 | US9597318, Code GK185)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301780(5-Phenyl-1-(thiazol-2-yl)pentan-1-one | US9597318...)copy SMILEScopy InChI
Affinity DataIC50: 3.05E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301781(4-(4-Octylphenoxy)-1-(thiazol-2-yl)butan-1-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.65E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301782(2-Fluoro-5-(4-(hexyloxy)phenyl)-1-(thiazol-2-yl)pe...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301777(US9597318, Code GK159)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301776(US9597318, Code GK152)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Avexxin AS

US Patent
LigandPNGBDBM301778(US9597318, Code GK160)copy SMILEScopy InChI
Affinity DataIC50: 7.20E+3nMAssay Description:Assay for cPLA2 activity was performed by the use of sonicated vesicles of 1-palmitoyl-2-arachidonoyl-sn-glycerol-3-phosphorylcholine (100 μM) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HH6N4CUS Patent