Compile Data Set for Download or QSAR
Found 35 Enz. Inhib. hit(s) with all data for assayid = 18 entry = 50010927
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543475(CHEMBL4649357)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543479(CHEMBL4639038)copy SMILEScopy InChI
Affinity DataIC50: 216nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543470(CHEMBL4634741)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543487(CHEMBL4634302)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543471(CHEMBL4639137)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543466(CHEMBL4647818)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543489(CHEMBL4648656)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543469(CHEMBL4637254)copy SMILEScopy InChI
Affinity DataIC50: 490nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543491(CHEMBL4645620)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543488(CHEMBL4646480)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543480(CHEMBL4641162)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543490(CHEMBL4644419)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543465(CHEMBL4636498)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543472(CHEMBL4647970)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543478(CHEMBL4644864)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543468(CHEMBL4637139)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543467(CHEMBL4636485)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543474(CHEMBL4645498)copy SMILEScopy InChI
Affinity DataIC50: 850nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543493(CHEMBL4649118)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543483(CHEMBL4643717)copy SMILEScopy InChI
Affinity DataIC50: 1.21E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543484(CHEMBL4633049)copy SMILEScopy InChI
Affinity DataIC50: 1.66E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543497(CHEMBL4649739)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543492(CHEMBL4636988)copy SMILEScopy InChI
Affinity DataIC50: 1.87E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543496(CHEMBL4644025)copy SMILEScopy InChI
Affinity DataIC50: 2.14E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543485(CHEMBL4647864)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543486(CHEMBL4649560)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543477(CHEMBL4643079)copy SMILEScopy InChI
Affinity DataIC50: 2.34E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543495(CHEMBL4641995)copy SMILEScopy InChI
Affinity DataIC50: 2.62E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543476(CHEMBL4647316)copy SMILEScopy InChI
Affinity DataIC50: 2.71E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543473(CHEMBL4638370)copy SMILEScopy InChI
Affinity DataIC50: 3.36E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543482(CHEMBL4632877)copy SMILEScopy InChI
Affinity DataIC50: 4.85E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543494(CHEMBL4638746)copy SMILEScopy InChI
Affinity DataIC50: 5.39E+3nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543498(CHEMBL4634971)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+4nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50158100(CHEMBL1614812)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+4nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed
TargetToll-like receptor 9(Homo sapiens (Human))
Princ

Curated by ChEMBL
LigandPNGBDBM50543481(CHEMBL4644144)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at human TLR9 overexpressed in HEK-Blue cells assessed as inhibition of ODN2006-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N55THPubMed