Compile Data Set for Download or QSAR
Found 15 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50005732
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407274(CHEMBL2111954)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed