Compile Data Set for Download or QSAR
Found 36 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50013981
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50014619(CHEMBL3184840)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50544742(CHEMBL4647910)copy SMILEScopy InChI
Affinity DataEC50:  63nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571376(CHEMBL4869477)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571377(CHEMBL4847403)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571378(CHEMBL4852570)copy SMILES
Affinity DataEC50:  5.57E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571379(CHEMBL4851385)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571380(CHEMBL4875648)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571381(CHEMBL4858793)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571382(CHEMBL4851809)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571383(CHEMBL4856959)copy SMILES
Affinity DataEC50:  3.75E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571384(CHEMBL4873660)copy SMILES
Affinity DataEC50:  2.71E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571385(CHEMBL4875417)copy SMILES
Affinity DataEC50:  705nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571386(CHEMBL4863277)copy SMILES
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571387(CHEMBL4857246)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571388(CHEMBL4846191)copy SMILES
Affinity DataEC50:  459nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571389(CHEMBL4863764)copy SMILES
Affinity DataEC50:  4.31E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571390(CHEMBL4849104)copy SMILES
Affinity DataEC50:  159nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571391(CHEMBL4864641)copy SMILES
Affinity DataEC50:  101nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571392(CHEMBL4857978)copy SMILES
Affinity DataEC50:  158nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571393(CHEMBL4850694)copy SMILES
Affinity DataEC50:  326nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571394(CHEMBL4861663)copy SMILES
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571395(CHEMBL4862328)copy SMILES
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571396(CHEMBL4865583)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571397(CHEMBL4856227)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571398(CHEMBL4865671)copy SMILES
Affinity DataEC50:  8.92E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571399(CHEMBL4866809)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571400(CHEMBL4859298)copy SMILES
Affinity DataEC50:  827nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571401(CHEMBL4867710)copy SMILES
Affinity DataEC50:  12nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571402(CHEMBL4851755)copy SMILES
Affinity DataEC50:  14nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571403(CHEMBL4850375)copy SMILES
Affinity DataEC50:  391nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571404(CHEMBL4854216)copy SMILES
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571405(CHEMBL4870280)copy SMILES
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571406(CHEMBL4876051)copy SMILES
Affinity DataEC50:  523nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50571407(CHEMBL4868247)copy SMILES
Affinity DataEC50:  2.32E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50183341(CHEMBL3817879)copy SMILEScopy InChI
Affinity DataEC50:  6.22E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed
TargetApelin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50544724(CHEMBL4641469)copy SMILEScopy InChI
Affinity DataEC50:  2.47E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RGNPubMed