Compile Data Set for Download or QSAR
Found 10 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50014960
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581547(CHEMBL5081349)copy SMILES
Affinity DataKi:  0.00736nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581544(CHEMBL5086475)copy SMILES
Affinity DataKi:  0.00826nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581548(CHEMBL5085124)copy SMILES
Affinity DataKi: <0.0100nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581546(CHEMBL5084416)copy SMILES
Affinity DataKi:  0.0114nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581549(CHEMBL5082483)copy SMILES
Affinity DataKi:  0.0370nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581542(CHEMBL5081587)copy SMILES
Affinity DataKi:  0.160nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581540(CHEMBL5087487)copy SMILES
Affinity DataKi:  0.230nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581537(CHEMBL5086286)copy SMILES
Affinity DataKi:  0.25nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581535(CHEMBL5091040)copy SMILES
Affinity DataKi:  0.390nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50581543(CHEMBL5094648)copy SMILES
Affinity DataKi:  2.30nMAssay Description:Inhibition of human PCSK9 using Alexa Fluor 674 as substrate incubated for 2 hrs by FRET plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7G0QPubMed