Compile Data Set for Download or QSAR
Found 14 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50034307
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360301(CHEMBL1933288 | US9150577, 93)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360293(CHEMBL1933280 | US9150577, 81)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360300(CHEMBL1933287 | US9150577, 105)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360291(CHEMBL1933278 | US9150577, 114)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360298(CHEMBL1933285 | US9150577, 53)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360302(CHEMBL1933289 | US9150577, 94)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360297(CHEMBL1933284)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360299(CHEMBL1933286 | US9150577, 54)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360294(CHEMBL1933281 | US9150577, 72)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360292(CHEMBL1933279 | US9150577, 64)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360296(CHEMBL1933283 | US9150577, 96)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360303(CHEMBL1933290 | US9150577, 99)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360290(CHEMBL1933277)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360295(CHEMBL1933282 | US9150577, 76)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed