TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 173nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Bristol Myers-Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
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