Compile Data Set for Download or QSAR
Found 11 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50047594
LigandPNGBDBM50398400(CHEMBL2178606)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177664(CHEMBL3814414)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177662(CHEMBL3813842)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50398399(CHEMBL2178608)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177666(CHEMBL3813906)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177668(CHEMBL3814925)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177669(CHEMBL3814544)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50358204(CHEMBL1922094)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177667(CHEMBL3815084)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177670(CHEMBL3814365)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed
LigandPNGBDBM50177671(CHEMBL3814933)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ05QDPubMed