Compile Data Set for Download or QSAR
Found 378 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 9912
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498332(US11014911, Example 157 | US11014911, Example 158 ...)copy SMILES
Affinity DataKi:  0.780nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498320(US11014911, Example 145 | US11718603, Example 145)copy SMILES
Affinity DataKi:  0.950nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498319(US11014911, Example 144 | US11718603, Example 144)copy SMILES
Affinity DataKi:  1.26nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498707((1R,3S)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  1.41nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498330(US11014911, Example 155 | US11014911, Example 156 ...)copy SMILES
Affinity DataKi:  1.63nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498334(US11014911, Example 159 | US11014911, Example 160 ...)copy SMILES
Affinity DataKi:  1.72nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498731((1S,3R)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  1.85nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498728((1S,3R)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  1.90nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498719((1S,3R)-3-(3-{[(2- methylpyridin-4- yl)acetyl]am...)copy SMILES
Affinity DataKi:  1.96nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498723((1S,3R)-3-(3-{[(6- methylpyridin-3- yl)acetyl]am...)copy SMILES
Affinity DataKi:  2.10nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498720((1S,3R)-3-(3-{[(6- methylpyridin-3- yl)acetyl]am...)copy SMILES
Affinity DataKi:  2.20nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498746((1S,3R)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.28nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498264(US11014911, Example 89 | US11014911, Example 90 | ...)copy SMILES
Affinity DataKi:  2.36nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498727((1S,3R)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.41nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498198(US11014911, Example 23 | US11718603, Example 23)copy SMILES
Affinity DataKi:  2.45nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498732((1S,3R)-3-(3-{[(5- methoxypyridin-2- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.60nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498802((1R,3S)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.76nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498796((1R,3S)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.77nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498234(US11014911, Example 59 | US11718603, Example 59)copy SMILES
Affinity DataKi:  2.89nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498726((1S,3R)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  2.94nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498707((1R,3S)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  2.97nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498725((1S,3R)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  3.12nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498724((1S,3R)-3-(3-{[(5- methylpyridin-2- yl)acetyl]am...)copy SMILES
Affinity DataKi:  3.24nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498745((1S,3R)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  3.29nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498822((1R,3S)-3-(3-{[(2-methoxy-1,3- thiazol-5-yl)acety...)copy SMILES
Affinity DataKi:  3.39nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498588((1R,3S)-3-(3-{[(1-methyl-1H- pyrazol-4-yl)acetyl]a...)copy SMILES
Affinity DataKi:  3.44nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498321(US11014911, Example 146 | US11718603, Example 146)copy SMILES
Affinity DataKi:  3.47nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498721((1S,3R)-3-(3-{[(5- methylpyridin-2- yl)acetyl]am...)copy SMILES
Affinity DataKi:  3.51nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498202(US11014911, Example 27 | US11718603, Example 27)copy SMILES
Affinity DataKi:  3.57nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498730((1S,3R)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  3.58nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498703((1R,3S)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  3.60nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498722((1S,3R)-3-(3-{[(2- methylpyridin-4- yl)acetyl]am...)copy SMILES
Affinity DataKi:  3.62nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498419((1R,3S)-3-(3-{[(6- methoxypyridin-3-yl) acetyl]a...)copy SMILES
Affinity DataKi:  3.70nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498709((1R,3S)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  3.80nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498326(US11014911, Example 151 | US11014911, Example 152 ...)copy SMILES
Affinity DataKi:  3.89nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498703((1R,3S)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  3.92nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498791((1R,3S)-3-(3-{[(6- methoxypyridin-3- yl)acetyl]a...)copy SMILES
Affinity DataKi:  4.05nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498740((1S,3R)-3-(3-{[(4- methoxyphenyl)acetyl]amino}- ...)copy SMILES
Affinity DataKi:  4.07nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498195(US11014911, Example 21 | US11718603, Example 21)copy SMILES
Affinity DataKi:  4.20nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498744((1S,3R)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  4.31nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498738((1S,3R)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  4.35nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498203(US11014911, Example 28 | US11718603, Example 28)copy SMILES
Affinity DataKi:  4.5nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498709((1R,3S)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  4.63nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498685((1S,3R)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl]...)copy SMILES
Affinity DataKi:  4.74nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498737((1S,3R)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl...)copy SMILES
Affinity DataKi:  4.85nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498184(US11014911, Example 12 | US11718603, Example 12)copy SMILES
Affinity DataKi:  4.86nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498250(US11014911, Example 75 | US11014911, Example 76 | ...)copy SMILES
Affinity DataKi:  4.96nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498800((1R,3S)-3-(3-{[(2- methoxypyridin-4- yl)acetyl]a...)copy SMILES
Affinity DataKi:  4.97nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498778((1R,3S)-3-(3-{[(3-methyl-1,2- oxazol-5-yl)acetyl]...)copy SMILES
Affinity DataKi:  5nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Pfizer Inc.

US Patent
LigandPNGBDBM498729((1S,3R)-3-(3-{[(5- methoxypyridin-2- yl)acetyl]a...)copy SMILES
Affinity DataKi:  5.11nMAssay Description:The purpose of GSK3β assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N26H2US Patent
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