Compile Data Set for Download or QSAR
Found 24 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50002504
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459401(CHEMBL4210854)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459392(CHEMBL4216873)copy SMILEScopy InChI
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459395(CHEMBL4210158)copy SMILEScopy InChI
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459396(CHEMBL4209266)copy SMILEScopy InChI
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459407(CHEMBL4204008)copy SMILEScopy InChI
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459394(CHEMBL4215258)copy SMILEScopy InChI
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50307118(5-[2-Chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-1...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459409(CHEMBL4218211)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459415(CHEMBL4206233)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459406(CHEMBL4213812)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459411(CHEMBL4206482)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459405(CHEMBL4205970)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459402(CHEMBL4202525)copy SMILEScopy InChI
Affinity DataKi:  82nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459403(CHEMBL4215696)copy SMILEScopy InChI
Affinity DataKi:  164nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459404(CHEMBL4205046)copy SMILEScopy InChI
Affinity DataKi:  239nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50177593((5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)...)copy SMILEScopy InChI
Affinity DataKi:  344nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459413(CHEMBL4218739)copy SMILEScopy InChI
Affinity DataKi:  504nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459410(CHEMBL4209421)copy SMILEScopy InChI
Affinity DataKi:  556nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459391(CHEMBL4209952)copy SMILEScopy InChI
Affinity DataKi:  573nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50094081((4-Amino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepi...)copy SMILEScopy InChI
Affinity DataKi:  734nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459393(CHEMBL4216926)copy SMILEScopy InChI
Affinity DataKi:  741nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459412(CHEMBL4207413)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459414(CHEMBL4207120)copy SMILEScopy InChI
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed