Compile Data Set for Download or QSAR
Found 13 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50011057
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101787(4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101782(4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101783(4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101781(4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101790(CHEMBL60334 | N-(4-Phenyl-thiazol-2-yl)-benzamide)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101786(2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101784(3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide | 4-...)copy SMILEScopy InChI
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101789(3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)copy SMILEScopy InChI
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101788(CHEMBL59978 | N-(4-Phenyl-thiazol-2-yl)-4-trifluor...)copy SMILEScopy InChI
Affinity DataKi:  165nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50101785(4-tert-Butyl-N-(4-phenyl-thiazol-2-yl)-benzamide |...)copy SMILEScopy InChI
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HM57QPPubMed