Found 16 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50012660 TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum AB
Curated by ChEMBL
Biovitrum AB
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
