Compile Data Set for Download or QSAR
Found 9 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50014387
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575511(CHEMBL4859677)copy SMILES
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575512(CHEMBL4854625)copy SMILES
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575513(CHEMBL4873903)copy SMILES
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575514(CHEMBL4852440)copy SMILES
Affinity DataEC50:  0.0370nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463446(US10781182, Compound IA2-142 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.937nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463447(US10781182, Compound IA2-143 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0630nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463443(US10781182, Compound IA2-120 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0360nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463445(US10781182, Compound IA2-140 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.233nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463444(US10781182, Compound IA2-121 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0350nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed