Compile Data Set for Download or QSAR
Found 27 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50015211
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583945(CHEMBL5080861)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50244495(CHEMBL4066176)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583942(CHEMBL5088454)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583946(CHEMBL5076817)copy SMILES
Affinity DataIC50: 59nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324284((R)-1-(tert-butyl)-N-(8-(2-((1-methyl-1H-pyrazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324285((R)-1-(tert-butyl)-N-(8-(2-((1-methyl-1H-pyrazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583947(CHEMBL5085931)copy SMILES
Affinity DataIC50: 104nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324290(5-(tert-butyl)-N-(2-(2-((1-methyl-1H-pyrazol-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583950(CHEMBL5094998)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50557487(Tolebrutinib)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324294(3-(tert-butyl)-N-(2-(2-((1-methyl-1H-pyrazol-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324293((R)-5-(tert-butyl)-N-(2-(2-((1-methyl-1H-pyrazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324337(5-(tert-butyl)-N-(2- (2-((1- methyl-1H-pyrazol-4- ...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583938(CHEMBL5090290)copy SMILES
Affinity DataIC50: 400nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583948(CHEMBL5081318)copy SMILES
Affinity DataIC50: 400nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583951(CHEMBL5073995)copy SMILES
Affinity DataIC50: 700nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324288((R)-1-(tert-butyl)-N-(2-(2-methoxyethyl)-8-(2-((1-...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM324380(1-(tert-butyl)-N- (2-(2-((1- methyl-1H-pyrazol-4- ...)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50369724(HM71224 | Ly3337641 | Poseltinib)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM291522(1-(4-(((6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50459553(CHEMBL4209441)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583930(CHEMBL5069979)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50194720(CHEMBL3900554)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583949(CHEMBL5075191)copy SMILES
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50553436(CHEMBL4744041)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed
TargetEarly activation antigen CD69(Homo sapiens)TBA
LigandPNGBDBM50583943(CHEMBL5083788)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CD69 in human whole blood preincubated for 30 mins followed by anti-human IgD stimulation and measured after 18 to 22 hrs by flow cytom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B641CPubMed