Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50018251
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50124215(CHEMBL3622866)copy SMILEScopy InChI
Affinity DataEC50:  200nMAssay Description:Antagonist activity at serotonin 5HT2A receptor assessed as effect on 5HT-induced isometric contractile force in isolated rings of pig coronary arter...More data for this Ligand-Target Pair
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50056695(CHEMBL3326918)copy SMILEScopy InChI
Affinity DataEC50:  3.23E+3nMAssay Description:Antagonist activity at serotonin 5HT2A receptor assessed as effect on 5HT-induced isometric contractile force in isolated rings of pig coronary arter...More data for this Ligand-Target Pair
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50056697(CHEMBL3326925)copy SMILEScopy InChI
Affinity DataEC50:  3.16E+3nMAssay Description:Antagonist activity at serotonin 5HT2A receptor assessed as effect on 5HT-induced isometric contractile force in isolated rings of pig coronary arter...More data for this Ligand-Target Pair
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50563775(CHEMBL4789165)copy SMILES
Affinity DataEC50:  1.96E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50563742(CHEMBL4795284)copy SMILES
Affinity DataEC50:  2.84E+4nMAssay Description:Antagonist activity at serotonin 5HT2A receptor assessed as effect on 5HT-induced isometric contractile force in isolated rings of pig coronary arter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50563743(CHEMBL4783434)copy SMILES
Affinity DataEC50:  2.48E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50056698(CHEMBL3326930)copy SMILEScopy InChI
Affinity DataEC50:  1.13E+3nMAssay Description:Antagonist activity at serotonin 5HT2A receptor assessed as effect on 5HT-induced isometric contractile force in isolated rings of pig coronary arter...More data for this Ligand-Target Pair
In DepthDetails