Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50025100
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
ActivX Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM15234((1R,3R,5S,9R,18S)-18-(methoxymethyl)-1,5-dimethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant Plk3 (unknown origin) assessed as casein substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M8XPubMed
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
ActivX Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of recombinant Plk3 (unknown origin) assessed as casein substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M8XPubMed