Compile Data Set for Download or QSAR
Found 10 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50027832
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265917(4-((4-tert-butylphenyl)ethynyl)benzoic acid | CHEM...)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265918(3-(4-((4-tert-butylphenyl)ethynyl)phenyl)-1,2,4-ox...)copy SMILEScopy InChI
Affinity DataEC50:  820nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265919(3-(3-((4-tert-butylphenyl)ethynyl)phenyl)-1,2,4-ox...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265920(4-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMedMMDB
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265949(3-(3-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronapht...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)copy SMILEScopy InChI
Affinity DataEC50:  8.60nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265950(5,5,8,8-tetramethyl-N-(4-(5-oxo-4,5-dihydro-1,2,4-...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265951(CHEMBL1657 | TAZAROTENE | US9963439, Tazarotene | ...)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMedDrugBank
TargetRetinoic acid receptor beta(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50265921(3-(4-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronapht...)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0TC9PubMed