Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50030371
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human neuromedin B receptor transfected in HEK293 cells assessed as inhibition of 1 nM neuromedin B-induced myo-[3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295236(11-(2-chloro-6-fluorophenyl)-3,3,8-trimethyl-2,3,4...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at human neuromedin B receptor transfected in HEK293 cells assessed as inhibition of 1 nM neuromedin B-induced myo-[3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed