Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50046188
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098420(CHEMBL3593411)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098416(CHEMBL3593407)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098414(CHEMBL3593247)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098418(CHEMBL3593409)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50322422(CHEMBL1173445 | Largazole)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098424(CHEMBL3593415)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098422(CHEMBL3593413)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098419(CHEMBL3593410)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098417(CHEMBL3593408)copy SMILEScopy InChI
Affinity DataIC50: 332nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098421(CHEMBL3593412)copy SMILEScopy InChI
Affinity DataIC50: 332nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098423(CHEMBL3593414)copy SMILEScopy InChI
Affinity DataIC50: 847nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Colorado State University

Curated by ChEMBL
LigandPNGBDBM50098415(CHEMBL3593406)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of recombinant full-length HDAC3 (unknown origin) using MAZ1600/MAZ1675 as substrate assessed as release of 7 amino-4-methylcoumarin measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP76QFPubMed