Compile Data Set for Download or QSAR
Found 38 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50047033
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145085(CHEMBL3763589)copy SMILEScopy InChI
Affinity DataEC50:  58nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataEC50:  3.60nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145090(CHEMBL3764811)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145091(CHEMBL3763164)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145092(CHEMBL3763531)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145093(CHEMBL3763661)copy SMILEScopy InChI
Affinity DataEC50:  6.70nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145094(CHEMBL3764422)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145095(CHEMBL3764670)copy SMILEScopy InChI
Affinity DataEC50:  8.5nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145096(CHEMBL3765611)copy SMILEScopy InChI
Affinity DataEC50:  6.10nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145097(CHEMBL3764829)copy SMILEScopy InChI
Affinity DataEC50:  41nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145098(CHEMBL3763844)copy SMILEScopy InChI
Affinity DataEC50:  9.5nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145099(CHEMBL3763243)copy SMILEScopy InChI
Affinity DataEC50:  9.70nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145100(CHEMBL3765318)copy SMILEScopy InChI
Affinity DataEC50:  23nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145101(CHEMBL3763674)copy SMILEScopy InChI
Affinity DataEC50:  3.80nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145131(CHEMBL3765291)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145132(CHEMBL3765434)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145133(CHEMBL3763188)copy SMILEScopy InChI
Affinity DataEC50:  18nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145134(CHEMBL3764464)copy SMILEScopy InChI
Affinity DataEC50:  24nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145135(CHEMBL3764188)copy SMILEScopy InChI
Affinity DataEC50:  9.30nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145136(CHEMBL3763963)copy SMILEScopy InChI
Affinity DataEC50:  27nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145137(CHEMBL3763370)copy SMILEScopy InChI
Affinity DataEC50:  121nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145138(CHEMBL3764085)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145139(CHEMBL3765125)copy SMILEScopy InChI
Affinity DataEC50:  149nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145142(CHEMBL3765056)copy SMILEScopy InChI
Affinity DataEC50:  6.90nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145143(CHEMBL3765528)copy SMILEScopy InChI
Affinity DataEC50:  5.5nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145148(CHEMBL3764990)copy SMILEScopy InChI
Affinity DataEC50:  285nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145149(CHEMBL3763822)copy SMILEScopy InChI
Affinity DataEC50:  6.90nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145150(CHEMBL3764066)copy SMILEScopy InChI
Affinity DataEC50:  164nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145151(CHEMBL3764202)copy SMILEScopy InChI
Affinity DataEC50:  18nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145152(CHEMBL3763446)copy SMILEScopy InChI
Affinity DataEC50:  5.10nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145153(CHEMBL3764624)copy SMILEScopy InChI
Affinity DataEC50:  250nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145154(CHEMBL3764920)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145155(CHEMBL3765670)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50084621(BMN 673 | Talazoparib)copy SMILEScopy InChI
Affinity DataEC50:  2.5nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145156(CHEMBL3764816)copy SMILEScopy InChI
Affinity DataEC50:  864nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataEC50:  5.90nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataEC50:  4.70nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145087(CHEMBL3764052)copy SMILEScopy InChI
Affinity DataEC50:  6nMAssay Description:Inhibition of PARP in human LoVo cells assessed as inhibition of poly(ADP)-ribose polymerization for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed