Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50005112
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
CIBA-GEIGY AG

Curated by ChEMBL
LigandPNGBDBM50032958(CHEMBL430501 | [3-Amino-2-(4-chloro-phenyl)-propyl...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58KDPPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
CIBA-GEIGY AG

Curated by ChEMBL
LigandPNGBDBM50032959(CHEMBL111378 | [3-Amino-2-(4-fluoro-phenyl)-propyl...)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58KDPPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
CIBA-GEIGY AG

Curated by ChEMBL
LigandPNGBDBM50032977((3-Amino-2-phenyl-propyl)-phosphinic acid | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58KDPPubMed