Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50006370
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)copy SMILEScopy InChI
Affinity DataKi:  201nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)copy SMILEScopy InChI
Affinity DataKi:  384nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)copy SMILEScopy InChI
Affinity DataKi:  833nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed