Compile Data Set for Download or QSAR
Found 41 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50012666
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559243(CHEMBL4794509)copy SMILES
Affinity DataIC50: 120nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 190nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354565(CHEMBL1836719)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559240(CHEMBL4755086)copy SMILES
Affinity DataIC50: 310nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559224(CHEMBL4788024)copy SMILES
Affinity DataIC50: 340nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559244(CHEMBL4753625)copy SMILES
Affinity DataIC50: 380nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559247(CHEMBL4789685)copy SMILES
Affinity DataIC50: 500nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559223(CHEMBL4788686)copy SMILES
Affinity DataIC50: 500nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559226(CHEMBL4754748)copy SMILES
Affinity DataIC50: 530nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559241(CHEMBL4739879)copy SMILES
Affinity DataIC50: 530nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559242(CHEMBL4748440)copy SMILES
Affinity DataIC50: 550nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559231(CHEMBL4792541)copy SMILES
Affinity DataIC50: 650nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354541(CHEMBL1836714)copy SMILEScopy InChI
Affinity DataIC50: 680nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559225(CHEMBL4763132)copy SMILES
Affinity DataIC50: 700nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559233(CHEMBL4753926)copy SMILES
Affinity DataIC50: 720nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559227(CHEMBL4748561)copy SMILES
Affinity DataIC50: 820nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559230(CHEMBL4783516)copy SMILES
Affinity DataIC50: 870nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559229(CHEMBL4745018)copy SMILES
Affinity DataIC50: 980nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559228(CHEMBL4788886)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559235(CHEMBL4760126)copy SMILES
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559246(CHEMBL4752999)copy SMILES
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559234(CHEMBL4781408)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354540(CHEMBL1836717)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559249(CHEMBL4753500)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559238(CHEMBL4793795)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559248(CHEMBL4759004)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354559(CHEMBL1836724)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559237(CHEMBL4747753)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559245(CHEMBL4740604)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559236(CHEMBL4796519)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559232(CHEMBL4740090)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559251(CHEMBL4756902)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559252(CHEMBL4754574)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559253(CHEMBL4763345)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559254(CHEMBL4745289)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354555(CHEMBL1836637)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559255(CHEMBL4761540)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559256(CHEMBL4782453)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559250(CHEMBL4799235)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559239(CHEMBL4794226)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed