Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50043684
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)copy SMILEScopy InChI
Affinity DataKi:  9.50E+4nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)copy SMILEScopy InChI
Affinity DataKi:  1.00E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)copy SMILEScopy InChI
Affinity DataKi:  1.07E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)copy SMILEScopy InChI
Affinity DataKi:  1.12E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)copy SMILEScopy InChI
Affinity DataKi:  1.21E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed