Compile Data Set for Download or QSAR
Found 8 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50046234
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102903(CHEMBL3394092)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102908(CHEMBL3393071)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50101585(CHEMBL3393986)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102904(CHEMBL3394091)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102872(CHEMBL3394083)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102878(CHEMBL3394082)copy SMILEScopy InChI
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed