Compile Data Set for Download or QSAR
Found 13 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50047692
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 5.88E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183562(CHEMBL3823599)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183450(CHEMBL3824133)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183451(CHEMBL3823551)copy SMILEScopy InChI
Affinity DataIC50: 3.03E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183563(CHEMBL3823697)copy SMILEScopy InChI
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183561(CHEMBL3824146)copy SMILEScopy InChI
Affinity DataIC50: 5.09E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183452(CHEMBL3824351)copy SMILEScopy InChI
Affinity DataIC50: 5.96E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183560(CHEMBL3822909)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183454(CHEMBL3822539)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183453(CHEMBL3824312)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183517(CHEMBL3823859 | US11773085, Compound B50)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed