TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.290nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Company, Ltd.
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
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