TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 237nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Oregon
Curated by ChEMBL
University of Oregon
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
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