Compile Data Set for Download or QSAR
Found 19 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50047788
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025042(CHEMBL3355105)copy SMILEScopy InChI
Affinity DataKi:  205nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025041(CHEMBL3355106)copy SMILEScopy InChI
Affinity DataKi:  241nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50190111(CHEMBL327844)copy SMILEScopy InChI
Affinity DataKi:  350nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50190110(CHEMBL254284)copy SMILEScopy InChI
Affinity DataKi:  1.03E+3nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)copy SMILEScopy InChI
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025047(CHEMBL3355100)copy SMILEScopy InChI
Affinity DataKi:  7.67E+3nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025048(CHEMBL3355099)copy SMILEScopy InChI
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50190113(CHEMBL3828715)copy SMILEScopy InChI
Affinity DataKi:  6.52E+4nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025049(CHEMBL3355107)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025050(CHEMBL3355108)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50025066(CHEMBL3355109)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170898(CHEMBL3805964)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50190109(Leucine Phosphonic acid)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170886(CHEMBL3804959)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50316049(1-amino-3-phenylpropylphosphonic acid | CHEMBL1090...)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170888(CHEMBL3805557)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170892(CHEMBL3804861)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170899(CHEMBL3806100)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50170895(CHEMBL3805487)copy SMILEScopy InChI
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SW1PubMed