Compile Data Set for Download or QSAR
Found 17 Enz. Inhib. hit(s) with all data for assayid = 7 entry = 50016185
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50166065((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataKi:  0.210nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50060070((S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phe...)copy SMILEScopy InChI
Affinity DataKi:  0.310nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50166054((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataKi:  0.350nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139015((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50166048((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139008((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139012((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | H-Tyr-Pro-Phe-Pro-NH2 | MORPHICEPTI...)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  104nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139019((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50068655(2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-butyryl]-1,2,3...)copy SMILEScopy InChI
Affinity DataKi:  167nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139009((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50166062((R)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.61E+3nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139016((R)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-1-oxo-prop...)copy SMILEScopy InChI
Affinity DataKi:  4.91E+3nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50139010((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  7.09E+3nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed