Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with all data for assayid = 8 entry = 50010529
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Eisai Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50079652((E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 17.2nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A1 receptor assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49Q0XPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Eisai Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A1 receptor assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49Q0XPubMed