Compile Data Set for Download or QSAR
Found 23 Enz. Inhib. hit(s) with all data for assayid = 8 entry = 50040373
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393218(CHEMBL1996510)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393214(CHEMBL2151411)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393228(CHEMBL2153750)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393219(CHEMBL2151415)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393229(CHEMBL2153751)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM33971(AEB071 | Sotrastaurin | med.21724, Compound 190)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393226(CHEMBL2153748)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393233(CHEMBL2153755)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393222(CHEMBL2151408)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393227(CHEMBL2153749)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393216(CHEMBL2151413)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393224(CHEMBL2151410)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393223(CHEMBL2151409)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393215(CHEMBL2151412)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM33970(maleimide derivative, 12)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393230(CHEMBL2153752)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393217(CHEMBL2151414)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393225(CHEMBL2153747)copy SMILEScopy InChI
Affinity DataIC50: 118nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393234(CHEMBL2153756)copy SMILEScopy InChI
Affinity DataIC50: 192nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393220(CHEMBL2151406)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393221(CHEMBL2151407)copy SMILEScopy InChI
Affinity DataIC50: 202nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393231(CHEMBL2153753)copy SMILEScopy InChI
Affinity DataIC50: 283nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50393232(CHEMBL2153754)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VR1PubMed