TargetProteasome subunit beta type-5(Homo sapiens (Human))
S£o Paulo State University
Curated by ChEMBL
S£o Paulo State University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human chymotrypsin-like activity of 20S proteasome (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of bacterial beta lactamase TEM-1More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of mouse liver HDAC using Boc-Lys (Ac)-AMC as substrate preincubated for 5 mins followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
S£o Paulo State University
Curated by ChEMBL
S£o Paulo State University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of full-length human recombinant PDE4B catalytic domain (152 to 484 residues)More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Selective estrogen receptor down regulator activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
S£o Paulo State University
Curated by ChEMBL
S£o Paulo State University
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human chymotrypsin-like activity of 20S proteasome (unknown origin)More data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium smegmatis (strain ATCC 700084 / mc(2...)TBA
Affinity DataIC50: 28nMAssay Description:Inhibition of mouse liver HDAC using Boc-Lys (Ac)-AMC as substrate preincubated for 5 mins followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human neutrophil ElastaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2C8(Homo sapiens (Human))
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP2C8 in human liver microsomes in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2B6(Homo sapiens (Human))
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP2B6 in human liver microsomes in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
TargetCytochrome P450 3A4(Homo sapiens (Human))
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
São Paulo State University (UNESP) , Institute of Chemistry, Araraquara 14800060, Brazil.
Curated by ChEMBL
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