TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University
Curated by ChEMBL
Semmelweis University
Curated by ChEMBL
Affinity DataIC50: 1.36E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway
Curated by ChEMBL
UiT - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
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