TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of rat PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant ACC2More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of c-Myc tagged human recombinant ACC2 expressed in baculovirus infected Sf9 cell system assessed as malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of human PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of human PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co, Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co, Ltd
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of rat ACC1More data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of rat ACC2More data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
TargetAcetyl-CoA carboxylase 1/2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human ACC1/2-mediated malonyl-CoA synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of human PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
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