TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP as substrate measured after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2KW5KKDPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2KW5KKDPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human PDE2 using c[8-3H]cAMP or c[8-3H]cGMP as substrate measured after 10 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.79E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.91E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.02E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.32E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.55E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 5.46E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Changzhou University
Curated by ChEMBL
Changzhou University
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of PDE2 (unknown origin) using [3H]cAMP or [3H]cGMP as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair