TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Compound was tested in vitro for binding affinity against Ionotropic glutamate receptor kainate using [3H]-kainate as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Compound was tested in vitro for binding affinity against mGluR1a metabotropic glutamate receptor, using [3H]-glutamate as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+5nMAssay Description:Compound was tested for its agonist activity against mGluR 2 receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+5nMAssay Description:Compound was tested for its agonist activity against mGluR 6 receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.15E+5nMAssay Description:Compound was tested in vitro for binding affinity against mGluR4a metabotropic glutamate receptor, using [3H]-L-AP4 as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Compound was tested for its antagonist activity against mGluR 2 receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+5nMAssay Description:Compound was tested in vitro for binding affinity against Ionotropic glutamate receptor AMPA, using [3H]-TCP as the radioligand.More data for this Ligand-Target Pair
Affinity DataEC50: >6.00E+5nMAssay Description:Compound was tested for its antagonist activity against mGluR 6 receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+5nMAssay Description:Compound was tested for its agonist activity against mGluR1a receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.05E+5nMAssay Description:Compound was tested for its agonist activity against mGluR 5a receptor in CHO cells.More data for this Ligand-Target Pair