TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 7.14nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 281nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 504nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 594nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 683nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.57E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [3H]-ZM-241,385 from A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 3.54E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 3.61E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 2.03E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 2.14E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 3.79E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 6.37E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 6.60E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.01E+5nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 1.07E+5nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 4.50E+3nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 6.80E+3nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 1.51E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 1.64E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 3.49E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 1.05E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 9.20E+3nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 3.20E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair