Compile Data Set for Download or QSAR
Found 269 of ki for UniProtKB: P32297
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50143314((+)-Epibatidine | (-)-epibatidine | (1R,2R,4S)-2-(...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK243 cell membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7ZBTPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49TF0PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Binding affinity to human alpha3beta4 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7N96PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)copy SMILEScopy InChI
Affinity DataKi:  0.457nMAssay Description:Binding affinity of the compound was determined against Nicotinic acetylcholine receptor using [3H]-(-)-nicotine radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8ZD0PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406472(CHEMBL4163848)copy SMILEScopy InChI
Affinity DataKi:  0.684nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406641(CHEMBL4170527)copy SMILEScopy InChI
Affinity DataKi:  0.799nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406541(CHEMBL4163257)copy SMILEScopy InChI
Affinity DataKi:  0.818nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406792(CHEMBL4174509)copy SMILEScopy InChI
Affinity DataKi:  0.988nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406686(CHEMBL4167298)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406544(CHEMBL4174940)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406500(CHEMBL4166573)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406685(CHEMBL4164252)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406539(CHEMBL4175573)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534298(CHEMBL4438684)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534286(CHEMBL4453542)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534287(CHEMBL4519018)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Binding affinity to alpha3beta4 nAChR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50500410(CHEMBL3745799)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534288(CHEMBL4472617)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50140291(CHEMBL3758455)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 nACh receptor expressed in HEK293 cells preincubated for 5 mins followed by radioligand addit...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2ZCHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406704(CHEMBL4160411)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Binding affinity to human alpha3beta4 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7N96PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534291(CHEMBL4559236)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534299(CHEMBL4450133)copy SMILEScopy InChI
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534300(CHEMBL4442125)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534284(CHEMBL4468804)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50538046(CHEMBL4647198)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534292(CHEMBL4437323)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406687(CHEMBL4164706)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50465459(CHEMBL4290888)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49TF0PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50465456(CHEMBL4283703)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49TF0PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM604954(US11667638, Example 160)copy SMILES
Affinity DataKi:  11.9nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VM4H7F
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534297(CHEMBL4443082)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406540(CHEMBL4177240)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534296(CHEMBL4557590)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)copy SMILES
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 transfected in HEK293 cell membranes preincubated for 5 mins followed by [3H]-epibatidine add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K93C4GPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534283(CHEMBL4440403)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534293(CHEMBL3341966)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H] epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50515321(CHEMBL4543232)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK243 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7ZBTPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534282(CHEMBL4437189)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406688(CHEMBL4166620)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50538045(CHEMBL4636163)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50515326(CHEMBL4565381)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK243 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7ZBTPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50203716(CHEMBL3982273)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-epibatine from human alpha3beta4-nACHR expressed in HEK243 cell membranes preincubated for 5 mins followed by overnight incubati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4MFRPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50140289(CHEMBL3759225)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 nACh receptor expressed in HEK293 cells preincubated for 5 mins followed by radioligand addit...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2ZCHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50597504(CHEMBL5177606)copy SMILES
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J96BDGPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM221048(US9284322, varenicline | US9303017, Varenicline)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50406538(CHEMBL4171125)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930WQMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50597507(CHEMBL5176101)copy SMILES
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J96BDGPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Istituto di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50534285(CHEMBL4453215)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QDQPubMed
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