Compile Data Set for Download or QSAR
Found 4 with your filter
TargetProtein tyrosine phosphatase type IVA 1(Homo sapiens (Human))TBA
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of full-length human brain His6-tagged PRL-1 expressed in Escherichia coli using TAMRA-Thr-Ala-Asp-Ile-Tyr(PO3H2)-Glu-NH2 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 1(Homo sapiens (Human))TBA
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant human His-6-tagged PTP4A1 expressed in Escherichia coli assessed as increase in polarization using TAMRAThr-Ala-Asp-Ile-Tyr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 1(Homo sapiens (Human))TBA
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Inhibition of full length human fusion His6 tagged PRL1 expressed in Escherichia coli using TAMRA-Thr-Ala-Asp-Ile-Tyr(PO3H2)-Glu-NH2 substrate by imm...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z8GPubMed
TargetProtein tyrosine phosphatase type IVA 1(Homo sapiens (Human))TBA
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of PRL1 (unknown origin) using DiFMUP as fluorogenic phosphate substrate assessed as DiFMUP dephosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z8GPubMed